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-Structure paper
Title | Structural Connection between Activation Microswitch and Allosteric Sodium Site in GPCR Signaling. |
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Journal, issue, pages | Structure, Vol. 26, Page 259-269.e5, Year 2018 |
Publish date | Jul 11, 2017 (structure data deposition date) |
Authors | White, K.L. / Eddy, M.T. / Gao, Z.G. / Han, G.W. / Lian, T. / Deary, A. / Patel, N. / Jacobson, K.A. / Katritch, V. / Stevens, R.C. |
External links | Structure / PubMed:29395784 |
Methods | X-ray diffraction |
Resolution | 2.6 - 2.9 Å |
Structure data | PDB-5wf5: PDB-5wf6: |
Chemicals | ChemComp-UKA: ChemComp-OLC: ChemComp-HOH: |
Source |
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Keywords | MEMBRANE PROTEIN / human A2a adenosine receptor / D52N / GPCR-T4L chimera / LCP / agonist / UK432097 / Activation microswitch / allosteric Na-site mutant / GPCR signaling / S91A |