+Search query
-Structure paper
Title | Discovery, Development, and Cellular Delivery of Potent and Selective Bicyclic Peptide Inhibitors of Grb7 Cancer Target. |
---|---|
Journal, issue, pages | J. Med. Chem., Vol. 60, Page 9349-9359, Year 2017 |
Publish date | Nov 20, 2016 (structure data deposition date) |
Authors | Watson, G.M. / Kulkarni, K. / Sang, J. / Ma, X. / Gunzburg, M.J. / Perlmutter, P. / Wilce, M.C.J. / Wilce, J.A. |
External links | J. Med. Chem. / PubMed:29083893 |
Methods | X-ray diffraction |
Resolution | 2.1 - 2.15 Å |
Structure data | PDB-5tyi: PDB-5u06: PDB-5u1q: |
Chemicals | ChemComp-HOH: ChemComp-K: ChemComp-CL: |
Source |
|
Keywords | Signaling Protein/Peptide / SH2 / inhibitor / bicyclic / Signaling Protein-Peptide complex / SIGNALING PROTEIN/INHIBITOR / Grb7 / SH2 domain / signalling / SIGNALING PROTEIN-PEPTIDE INHIBITOR complex / SIGNALING PROTEIN-INHIBITOR complex / SIGNALING PROTEIN/PEPTIDE INHIBITOR |