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-Structure paper
Title | Discovery of Potent and Selective Inhibitors for G9a-Like Protein (GLP) Lysine Methyltransferase. |
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Journal, issue, pages | J. Med. Chem., Vol. 60, Page 1876-1891, Year 2017 |
Publish date | Nov 3, 2016 (structure data deposition date) |
![]() | Xiong, Y. / Li, F. / Babault, N. / Dong, A. / Zeng, H. / Wu, H. / Chen, X. / Arrowsmith, C.H. / Brown, P.J. / Liu, J. ...Xiong, Y. / Li, F. / Babault, N. / Dong, A. / Zeng, H. / Wu, H. / Chen, X. / Arrowsmith, C.H. / Brown, P.J. / Liu, J. / Vedadi, M. / Jin, J. |
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Methods | X-ray diffraction |
Resolution | 1.66 - 2.6 Å |
Structure data | ![]() PDB-5ttf: ![]() PDB-5ttg: ![]() PDB-5tuy: ![]() PDB-5tuz: |
Chemicals | ![]() ChemComp-ZN: ![]() ChemComp-SAM: ![]() ChemComp-7KZ: ![]() ChemComp-CL: ![]() ChemComp-UNX: ![]() ChemComp-HOH: ![]() ChemComp-GOL: ![]() ChemComp-DMS: ![]() ChemComp-7L6: ![]() ChemComp-EDO: |
Source |
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![]() | TRANSFERASE / EHMT2 / G9a / BAT8 / methyltransferase / UNC3832 / Structural Genomics / Structural Genomics Consortium / SGC / EHMT1 / GLP / MS012 / TRANSFERASE/TRANSFERASE INHIBITOR / Methyl-TRANSFERASE INHIBITOR complex / TRANSFERASE-TRANSFERASE INHIBITOR complex / Methyl Transferase |