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-Structure paper
タイトル | Structure-based design and mechanisms of allosteric inhibitors for mitochondrial branched-chain alpha-ketoacid dehydrogenase kinase. |
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ジャーナル・号・ページ | Proc. Natl. Acad. Sci. USA, Vol. 110, Page 9728-9733, Year 2013 |
掲載日 | 2011年9月26日 (構造データの登録日) |
![]() | Tso, S.C. / Qi, X. / Gui, W.J. / Chuang, J.L. / Morlock, L.K. / Wallace, A.L. / Ahmed, K. / Laxman, S. / Campeau, P.M. / Lee, B.H. ...Tso, S.C. / Qi, X. / Gui, W.J. / Chuang, J.L. / Morlock, L.K. / Wallace, A.L. / Ahmed, K. / Laxman, S. / Campeau, P.M. / Lee, B.H. / Hutson, S.M. / Tu, B.P. / Williams, N.S. / Tambar, U.K. / Wynn, R.M. / Chuang, D.T. |
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手法 | X線回折 |
解像度 | 2.05 - 2.85 Å |
構造データ | ![]() PDB-3tz0: ![]() PDB-3tz2: ![]() PDB-3tz4: ![]() PDB-3tz5: ![]() PDB-4dzy: ![]() PDB-4h7q: ![]() PDB-4h81: ![]() PDB-4h85: |
化合物 | ![]() ChemComp-03H: ![]() ChemComp-HOH: ![]() ChemComp-CLT: ![]() ChemComp-ADP: ![]() ChemComp-MG: ![]() ChemComp-K: ![]() ChemComp-WJ1: ![]() ChemComp-COI: ![]() ChemComp-WJ2: ![]() ChemComp-HRI: |
由来 |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / GHKL protein kinase / Allosteric kinase inhibitor / Branched-chain alpha-ketoacid / Branched-chain amino acids / Maple syrup urine disease / Diabetes and obesity / Bergerat nucleotide-binding fold / Protein kinase / TRANSFERASE-TRANSFERASE INHIBITOR complex / transferase |