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-Structure paper
Title | Sinefungin Derivatives as Inhibitors and Structure Probes of Protein Lysine Methyltransferase SETD2. |
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Journal, issue, pages | J. Am. Chem. Soc., Vol. 134, Page 18004-18014, Year 2012 |
Publish date | Jun 18, 2012 (structure data deposition date) |
![]() | Zheng, W. / Ibanez, G. / Wu, H. / Blum, G. / Zeng, H. / Dong, A. / Li, F. / Hajian, T. / Allali-Hassani, A. / Amaya, M.F. ...Zheng, W. / Ibanez, G. / Wu, H. / Blum, G. / Zeng, H. / Dong, A. / Li, F. / Hajian, T. / Allali-Hassani, A. / Amaya, M.F. / Siarheyeva, A. / Yu, W. / Brown, P.J. / Schapira, M. / Vedadi, M. / Min, J. / Luo, M. |
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Methods | X-ray diffraction |
Resolution | 2.06 - 2.1 Å |
Structure data | ![]() PDB-4fmu: ![]() PDB-4h12: |
Chemicals | ![]() ChemComp-ZN: ![]() ChemComp-0UM: ![]() ChemComp-UNX: ![]() ChemComp-HOH: ![]() ChemComp-SAH: ![]() ChemComp-CL: |
Source |
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![]() | TRANSFERASE / Structural Genomics Consortium / SGC / Methyltransferase / SET domain-containing protein 2 / Pr-SNF / S-adenosyl-L-homocysteine / structural genomics / activator / chromatin regulator / DNA-binding / methylation / nucleus / phosphoprotein / transcription / transcription regulation |