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-Structure paper
| Title | Structure of human G protein-coupled receptor kinase 2 in complex with the kinase inhibitor balanol. |
|---|---|
| Journal, issue, pages | J. Med. Chem., Vol. 53, Page 1867-1870, Year 2010 |
| Publish date | Mar 11, 2008 (structure data deposition date) |
Authors | Tesmer, J.J. / Tesmer, V.M. / Lodowski, D.T. / Steinhagen, H. / Huber, J. |
External links | J. Med. Chem. / PubMed:20128603 |
| Methods | X-ray diffraction |
| Resolution | 2.75 - 3.1 Å |
| Structure data | ![]() PDB-3cik: ![]() PDB-3krw: ![]() PDB-3krx: |
| Chemicals | ![]() ChemComp-MG: ![]() ChemComp-HOH: ![]() ChemComp-BA1: |
| Source |
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Keywords | Transferase/Signaling protein / protein kinase / complex / G protein / receptor / WD40 repeat / ATP-binding / Nucleotide-binding / Serine/threonine-protein kinase / Transferase / Transducer / WD repeat / Lipoprotein / Membrane / Phosphoprotein / Prenylation / Transferase-Signaling protein COMPLEX / PROTEIN BINDING / INHIBITOR / WD40 / PH DOMAIN / RGS HOMOLOGY DOMAIN / Kinase / Polymorphism / Acetylation / Cell membrane / Methylation |
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homo sapiens (human)
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