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-Structure paper
Title | Flavopiridol inhibits glycogen phosphorylase by binding at the inhibitor site. |
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Journal, issue, pages | J. Biol. Chem., Vol. 275, Page 34566-34573, Year 2000 |
Publish date | May 11, 2000 (structure data deposition date) |
Authors | Oikonomakos, N.G. / Schnier, J.B. / Zographos, S.E. / Skamnaki, V.T. / Tsitsanou, K.E. / Johnson, L.N. |
External links | J. Biol. Chem. / PubMed:10924512 |
Methods | X-ray diffraction |
Resolution | 1.76 - 2.3 Å |
Structure data | PDB-1c8k: PDB-1e1y: PDB-1gfz: |
Chemicals | ChemComp-PLP: ChemComp-CPB: ChemComp-HOH: ChemComp-PO3: ChemComp-GLC: ChemComp-IMP: ChemComp-CFF: |
Source |
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Keywords | TRANSFERASE / GLYCOGEN METABOLISM / GLYCOGEN PHOSPHORYLASE B / INHIBITION / INHIBITOR BINDING SITE / ANTITUMOUR AGENT / ALLOSTERIC INHIBITION / GLYCOGEN PHOSPHORYLASE / DIABETES / FLAVOPIRIDOL / INHIBITOR SITE |