- PDB-8uwn: Crystal structure of human CLK1 kinase in complex with compound 3 -
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基本情報
登録情報
データベース: PDB / ID: 8uwn
タイトル
Crystal structure of human CLK1 kinase in complex with compound 3
要素
Dual specificity protein kinase CLK1
キーワード
SIGNALING PROTEIN / Kinase / Inhibitor / Transferase
機能・相同性
機能・相同性情報
dual-specificity kinase / regulation of RNA splicing / protein serine/threonine/tyrosine kinase activity / non-membrane spanning protein tyrosine kinase activity / protein tyrosine kinase activity / protein serine kinase activity / protein serine/threonine kinase activity / ATP binding / nucleus 類似検索 - 分子機能
: / Serine/threonine-protein kinase, active site / Serine/Threonine protein kinases active-site signature. / Protein kinase domain / Serine/Threonine protein kinases, catalytic domain / Protein kinase, ATP binding site / Protein kinases ATP-binding region signature. / Protein kinase domain profile. / Protein kinase domain / Protein kinase-like domain superfamily 類似検索 - ドメイン・相同性
: / Dual specificity protein kinase CLK1 類似検索 - 構成要素
構造決定の手法: 分子置換 / 解像度: 1.8→29.35 Å / Cor.coef. Fo:Fc: 0.962 / Cor.coef. Fo:Fc free: 0.925 / SU B: 4.016 / SU ML: 0.116 / 交差検証法: THROUGHOUT / ESU R: 0.132 / ESU R Free: 0.139 / 立体化学のターゲット値: MAXIMUM LIKELIHOOD / 詳細: HYDROGENS HAVE BEEN ADDED IN THE RIDING POSITIONS
Rfactor
反射数
%反射
Selection details
Rfree
0.24034
1864
4.9 %
RANDOM
Rwork
0.17709
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obs
0.18015
35813
97.78 %
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溶媒の処理
イオンプローブ半径: 0.8 Å / 減衰半径: 0.8 Å / VDWプローブ半径: 1.2 Å / 溶媒モデル: BABINET MODEL WITH MASK