登録情報 | データベース: PDB / ID: 8qb2 |
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タイトル | Crystal Structure of BRPF1 bromodomain in complex with acetyl-pyrrole derivative compound 79 |
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要素 | Peregrin |
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キーワード | TRANSCRIPTION / four helical bundle |
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機能・相同性 | 機能・相同性情報
acetyltransferase activator activity / regulation of developmental process / regulation of hemopoiesis / MOZ/MORF histone acetyltransferase complex / histone acetyltransferase complex / Regulation of TP53 Activity through Acetylation / HATs acetylate histones / chromatin remodeling / regulation of DNA-templated transcription / regulation of transcription by RNA polymerase II ...acetyltransferase activator activity / regulation of developmental process / regulation of hemopoiesis / MOZ/MORF histone acetyltransferase complex / histone acetyltransferase complex / Regulation of TP53 Activity through Acetylation / HATs acetylate histones / chromatin remodeling / regulation of DNA-templated transcription / regulation of transcription by RNA polymerase II / positive regulation of DNA-templated transcription / DNA binding / nucleoplasm / nucleus / metal ion binding / plasma membrane / cytosol / cytoplasm類似検索 - 分子機能 BRPF1, PHD domain / Peregrin, ePHD domain / : / : / Enhancer of polycomb-like, N-terminal / Enhancer of polycomb-like / PHD-finger / PHD-zinc-finger like domain / Extended PHD (ePHD) domain / Extended PHD (ePHD) domain profile. ...BRPF1, PHD domain / Peregrin, ePHD domain / : / : / Enhancer of polycomb-like, N-terminal / Enhancer of polycomb-like / PHD-finger / PHD-zinc-finger like domain / Extended PHD (ePHD) domain / Extended PHD (ePHD) domain profile. / domain with conserved PWWP motif / PWWP domain / PWWP domain profile. / PWWP domain / Zinc finger C2H2 type domain profile. / Zinc finger, PHD-type, conserved site / Zinc finger C2H2 type domain signature. / Zinc finger PHD-type signature. / Zinc finger C2H2-type / Zinc finger PHD-type profile. / Zinc finger, PHD-finger / Zinc finger, PHD-type / PHD zinc finger / Zinc finger, FYVE/PHD-type / Bromodomain, conserved site / Bromodomain signature. / Bromodomain / Bromodomain profile. / bromo domain / Bromodomain / Bromodomain-like superfamily / Zinc finger, RING/FYVE/PHD-type類似検索 - ドメイン・相同性 |
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生物種 | Homo sapiens (ヒト) |
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手法 | X線回折 / シンクロトロン / 分子置換 / 解像度: 1.42 Å |
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データ登録者 | Dalle Vedove, A. / Cazzanelli, G. / Lolli, G. |
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資金援助 | イタリア, 1件 組織 | 認可番号 | 国 |
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Italian Association for Cancer Research | MFAG 2017 - ID. 19882 | イタリア |
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引用 | ジャーナル: To be published タイトル: Dual BET/BRPF1 inhibitors induce morphological alteration and cellular death in various human cancer cell lines 著者: Cazzanelli, G. / Dalle Vedove, A. / Caflisch, A. / Lolli, G. |
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履歴 | 登録 | 2023年8月24日 | 登録サイト: PDBE / 処理サイト: PDBE |
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改定 1.0 | 2024年9月11日 | Provider: repository / タイプ: Initial release |
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