登録情報 | データベース: PDB / ID: 6ibb |
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タイトル | Crystal structure of the rat isoform of the succinate receptor SUCNR1 (GPR91) in complex with a nanobody |
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要素 | - Nanobody6
- Succinate receptor 1
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キーワード | MEMBRANE PROTEIN / SUCNR1 GPR91 GPCR G-Protein coupled receptor Nanobody Succinate Complex |
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機能・相同性 | 機能・相同性情報
Class A/1 (Rhodopsin-like receptors) / regulation of angiotensin metabolic process / renin secretion into blood stream / positive regulation of chemotaxis / macrophage activation involved in immune response / G alpha (i) signalling events / G protein-coupled receptor activity / response to calcium ion / positive regulation of inflammatory response / glucose homeostasis ...Class A/1 (Rhodopsin-like receptors) / regulation of angiotensin metabolic process / renin secretion into blood stream / positive regulation of chemotaxis / macrophage activation involved in immune response / G alpha (i) signalling events / G protein-coupled receptor activity / response to calcium ion / positive regulation of inflammatory response / glucose homeostasis / signaling receptor activity / G protein-coupled receptor signaling pathway / plasma membrane類似検索 - 分子機能 G-protein coupled receptors family 1 signature. / G protein-coupled receptor, rhodopsin-like / GPCR, rhodopsin-like, 7TM / G-protein coupled receptors family 1 profile. / 7 transmembrane receptor (rhodopsin family)類似検索 - ドメイン・相同性 CHOLESTEROL / (2~{S},5~{R})-hexane-2,5-diol / (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate / Succinate receptor 1類似検索 - 構成要素 |
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生物種 | Rattus norvegicus (ドブネズミ) Vicugna pacos (アルパカ) |
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手法 | X線回折 / シンクロトロン / 分子置換 / 解像度: 2.12 Å |
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データ登録者 | Haffke, M. / Jaakola, V.-P. |
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引用 | ジャーナル: Nature / 年: 2019 タイトル: Structural basis of species-selective antagonist binding to the succinate receptor. 著者: Haffke, M. / Fehlmann, D. / Rummel, G. / Boivineau, J. / Duckely, M. / Gommermann, N. / Cotesta, S. / Sirockin, F. / Freuler, F. / Littlewood-Evans, A. / Kaupmann, K. / Jaakola, V.P. |
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履歴 | 登録 | 2018年11月29日 | 登録サイト: PDBE / 処理サイト: PDBE |
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改定 1.0 | 2019年8月14日 | Provider: repository / タイプ: Initial release |
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改定 1.1 | 2019年10月16日 | Group: Data collection / Database references / カテゴリ: citation Item: _citation.country / _citation.journal_abbrev ..._citation.country / _citation.journal_abbrev / _citation.journal_id_ASTM / _citation.journal_id_CSD / _citation.journal_id_ISSN / _citation.pdbx_database_id_DOI / _citation.title / _citation.year |
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改定 1.2 | 2019年11月6日 | Group: Data collection / Database references / カテゴリ: citation / citation_author Item: _citation.journal_volume / _citation.page_first ..._citation.journal_volume / _citation.page_first / _citation.page_last / _citation.pdbx_database_id_PubMed / _citation.title |
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改定 1.3 | 2024年1月24日 | Group: Data collection / Database references / Refinement description カテゴリ: chem_comp_atom / chem_comp_bond ...chem_comp_atom / chem_comp_bond / database_2 / pdbx_initial_refinement_model Item: _database_2.pdbx_DOI / _database_2.pdbx_database_accession |
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