Entry Database : PDB / ID : 5x72 Structure visualization Downloads & linksTitle The crystal Structure PDE delta in complex with (rac)-p9 ComponentsRetinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit delta Details Keywords LIPID BINDING PROTEINFunction / homology Function and homology informationFunction Domain/homology Component
ARL13B-mediated ciliary trafficking of INPP5E / GTPase inhibitor activity / response to stimulus / visual perception / cytoplasmic vesicle membrane / cilium / small GTPase binding / RAS processing / cytoplasmic vesicle / cytoskeleton ... ARL13B-mediated ciliary trafficking of INPP5E / GTPase inhibitor activity / response to stimulus / visual perception / cytoplasmic vesicle membrane / cilium / small GTPase binding / RAS processing / cytoplasmic vesicle / cytoskeleton / cytosol / cytoplasm Similarity search - Function GMP phosphodiesterase, delta subunit / Retinal rod rhodopsin-sensitive cGMP 3', 5'-cyclic phosphodiesterase, delta subunit / GMP phosphodiesterase, delta subunit / GMP phosphodiesterase, delta subunit superfamily / GMP-PDE, delta subunit / Coagulation Factor XIII; Chain A, domain 1 / Distorted Sandwich / Immunoglobulin E-set / Mainly Beta Similarity search - Domain/homologyBiological species Homo sapiens (human)Method X-RAY DIFFRACTION / SYNCHROTRON / MOLECULAR REPLACEMENT / Resolution : 1.95 Å DetailsAuthors Jiang, Y. / Zhuang, C. / Chen, L. / Wang, R. / Wang, F. / Sheng, C. Funding support China, 1items Details Hide detailsOrganization Grant number Country National Basic Research Program of China 2014CB541800 China
CitationJournal : J. Med. Chem. / Year : 2017Title : Structural Biology-Inspired Discovery of Novel KRAS-PDE delta InhibitorsAuthors : Jiang, Y. / Zhuang, C. / Chen, L. / Lu, J. / Dong, G. / Miao, Z. / Zhang, W. / Li, J. / Sheng, C. History Deposition Feb 23, 2017 Deposition site : PDBJ / Processing site : PDBJRevision 1.0 Oct 4, 2017 Provider : repository / Type : Initial releaseRevision 1.1 Dec 6, 2017 Group : Database references / Category : citationItem : _citation.journal_volume / _citation.page_first / _citation.page_lastRevision 1.2 Nov 22, 2023 Group : Data collection / Database references / Refinement descriptionCategory : chem_comp_atom / chem_comp_bond ... chem_comp_atom / chem_comp_bond / database_2 / pdbx_initial_refinement_model Item : _database_2.pdbx_DOI / _database_2.pdbx_database_accession
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