登録情報 | データベース: PDB / ID: 5nra |
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タイトル | Crystal structure of human chitotriosidase-1 (hCHIT) catalytic domain in complex with compound 7g |
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要素 | Chitotriosidase-1 |
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キーワード | HYDROLASE / chitotriosidase-1 (hCHIT) catalytic domain in complex with compound 7g |
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機能・相同性 | 機能・相同性情報
endochitinase activity / polysaccharide digestion / Digestion of dietary carbohydrate / chitinase / chitinase activity / chitin catabolic process / chitin binding / polysaccharide catabolic process / hydrolase activity, hydrolyzing O-glycosyl compounds / response to bacterium ...endochitinase activity / polysaccharide digestion / Digestion of dietary carbohydrate / chitinase / chitinase activity / chitin catabolic process / chitin binding / polysaccharide catabolic process / hydrolase activity, hydrolyzing O-glycosyl compounds / response to bacterium / specific granule lumen / tertiary granule lumen / lysosome / immune response / Neutrophil degranulation / extracellular space / extracellular region類似検索 - 分子機能 Chitin-binding domain type 2 / Chitin binding domain / Chitin binding Peritrophin-A domain / Chitin-binding type-2 domain profile. / Chitin binding domain superfamily / Glycosyl hydrolases family 18 (GH18) active site / Glycosyl hydrolases family 18 (GH18) active site signature. / : / Chitinase insertion domain superfamily / Chitinase II ...Chitin-binding domain type 2 / Chitin binding domain / Chitin binding Peritrophin-A domain / Chitin-binding type-2 domain profile. / Chitin binding domain superfamily / Glycosyl hydrolases family 18 (GH18) active site / Glycosyl hydrolases family 18 (GH18) active site signature. / : / Chitinase insertion domain superfamily / Chitinase II / Glyco_18 / Glycosyl hydrolases family 18 (GH18) domain profile. / Glycosyl hydrolases family 18 / Glycoside hydrolase family 18, catalytic domain / Glycoside hydrolase superfamily類似検索 - ドメイン・相同性 |
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生物種 | Homo sapiens (ヒト) |
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手法 | X線回折 / シンクロトロン / 分子置換 / 解像度: 1.267 Å |
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データ登録者 | Mazur, M. / Olczak, J. / Olejniczak, S. / Koralewski, R. / Czestkowski, W. / Jedrzejczak, A. / Golab, J. / Dzwonek, K. / Dymek, B. / Sklepkiewicz, P. ...Mazur, M. / Olczak, J. / Olejniczak, S. / Koralewski, R. / Czestkowski, W. / Jedrzejczak, A. / Golab, J. / Dzwonek, K. / Dymek, B. / Sklepkiewicz, P. / Zagozdzon, A. / Noonan, T. / Mahboubi, K. / Conway, B. / Sheeler, R. / Beckett, P. / Hungerford, W.M. / Podjarny, A. / Mitschler, A. / Cousido-Siah, A. / Fadel, F. / Golebiowski, A. |
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引用 | ジャーナル: J. Med. Chem. / 年: 2018 タイトル: Targeting Acidic Mammalian chitinase Is Effective in Animal Model of Asthma. 著者: Mazur, M. / Olczak, J. / Olejniczak, S. / Koralewski, R. / Czestkowski, W. / Jedrzejczak, A. / Golab, J. / Dzwonek, K. / Dymek, B. / Sklepkiewicz, P.L. / Zagozdzon, A. / Noonan, T. / ...著者: Mazur, M. / Olczak, J. / Olejniczak, S. / Koralewski, R. / Czestkowski, W. / Jedrzejczak, A. / Golab, J. / Dzwonek, K. / Dymek, B. / Sklepkiewicz, P.L. / Zagozdzon, A. / Noonan, T. / Mahboubi, K. / Conway, B. / Sheeler, R. / Beckett, P. / Hungerford, W.M. / Podjarny, A. / Mitschler, A. / Cousido-Siah, A. / Fadel, F. / Golebiowski, A. |
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履歴 | 登録 | 2017年4月22日 | 登録サイト: PDBE / 処理サイト: PDBE |
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改定 1.0 | 2018年3月28日 | Provider: repository / タイプ: Initial release |
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改定 1.1 | 2019年10月16日 | Group: Data collection / カテゴリ: reflns_shell |
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改定 1.2 | 2024年1月17日 | Group: Advisory / Data collection ...Advisory / Data collection / Database references / Refinement description カテゴリ: chem_comp_atom / chem_comp_bond ...chem_comp_atom / chem_comp_bond / database_2 / pdbx_initial_refinement_model / pdbx_unobs_or_zero_occ_atoms Item: _database_2.pdbx_DOI / _database_2.pdbx_database_accession |
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