- PDB-4uf0: Crystal structure of JmjC domain of human histone demethylase UTY... -
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IDまたはキーワード:
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基本情報
登録情報
データベース: PDB / ID: 4uf0
タイトル
Crystal structure of JmjC domain of human histone demethylase UTY in complex with epitherapuetic compound 2-(((2-((2-(dimethylamino)ethyl) (ethyl)amino)-2-oxoethyl)amino)methyl)isonicotinic acid.
要素
(HISTONE DEMETHYLASE ...) x 2
キーワード
OXIDOREDUCTASE
機能・相同性
機能・相同性情報
[histone H3]-trimethyl-L-lysine27 demethylase / histone H3K27me2/H3K27me3 demethylase activity / MLL3/4 complex / histone demethylase activity / HDMs demethylate histones / chromatin DNA binding / heart development / regulation of gene expression / RNA polymerase II cis-regulatory region sequence-specific DNA binding / nucleoplasm / metal ion binding 類似検索 - 分子機能
HISTONEDEMETHYLASEUTY / UBIQUITOUSLY-TRANSCRIBED TPR PROTEIN ON THE Y CHROMOSOME / UBIQUITOUSLY-TRANSCRIBED Y CHROMOSOME ...UBIQUITOUSLY-TRANSCRIBED TPR PROTEIN ON THE Y CHROMOSOME / UBIQUITOUSLY-TRANSCRIBED Y CHROMOSOME TETRATRICOPEPTIDE REPEAT PROTEIN
HISTONEDEMETHYLASEUTY / UBIQUITOUSLY-TRANSCRIBED TPR PROTEIN ON THE Y CHROMOSOME / UBIQUITOUSLY-TRANSCRIBED Y CHROMOSOME ...UBIQUITOUSLY-TRANSCRIBED TPR PROTEIN ON THE Y CHROMOSOME / UBIQUITOUSLY-TRANSCRIBED Y CHROMOSOME TETRATRICOPEPTIDE REPEAT PROTEIN
5,6-DIHYDRO-BENZO[H]CINNOLIN-3-YLAMINE (MMK): DIMETHYLAMINE GROUP DID NOT SHOW ANY DENSITY SO ...5,6-DIHYDRO-BENZO[H]CINNOLIN-3-YLAMINE (MMK): DIMETHYLAMINE GROUP DID NOT SHOW ANY DENSITY SO REFINED WITH ZERO OCCUPANCY
解像度: 1.78→81.03 Å / Cor.coef. Fo:Fc: 0.972 / Cor.coef. Fo:Fc free: 0.953 / SU B: 5.892 / SU ML: 0.08 / 交差検証法: THROUGHOUT / ESU R: 0.118 / ESU R Free: 0.103 / 立体化学のターゲット値: MAXIMUM LIKELIHOOD 詳細: U VALUES REFINED INDIVIDUALLY DIMETHYLAMINE GROUP OF THE DRG LIGAND OCCUPANCY WAS SET UP TO ZERO AS WE DO NOT SEE ANY DENSITY
Rfactor
反射数
%反射
Selection details
Rfree
0.21517
5650
4.9 %
RANDOM
Rwork
0.14857
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obs
0.15184
109117
99.97 %
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溶媒の処理
イオンプローブ半径: 0.8 Å / 減衰半径: 0.8 Å / VDWプローブ半径: 1.2 Å / 溶媒モデル: MASK