Entry | Database: PDB / ID: 4cax |
---|
Title | Crystal structure of Aspergillus fumigatus N-myristoyl transferase in complex with myristoyl CoA and a pyrazole sulphonamide ligand (DDD85646) |
---|
Components | GLYCYLPEPTIDE N-TETRADECANOYLTRANSFERASE |
---|
Keywords | TRANSFERASE / DRUG DISCOVERY |
---|
Function / homology | Function and homology information
glycylpeptide N-tetradecanoyltransferase / glycylpeptide N-tetradecanoyltransferase activity / cytoplasm / cytosolSimilarity search - Function Glycylpeptide N-tetradecanoyltransferase, conserved site / Myristoyl-CoA:protein N-myristoyltransferase signature 1. / Myristoyl-CoA:protein N-myristoyltransferase signature 2. / Glycylpeptide N-tetradecanoyltransferase / Glycylpeptide N-tetradecanoyltransferase, N-terminal / Glycylpeptide N-tetradecanoyltransferase, C-terminal / Myristoyl-CoA:protein N-myristoyltransferase, N-terminal domain / Myristoyl-CoA:protein N-myristoyltransferase, C-terminal domain / Gcn5-related N-acetyltransferase (GNAT) / Acyl-CoA N-acyltransferase ...Glycylpeptide N-tetradecanoyltransferase, conserved site / Myristoyl-CoA:protein N-myristoyltransferase signature 1. / Myristoyl-CoA:protein N-myristoyltransferase signature 2. / Glycylpeptide N-tetradecanoyltransferase / Glycylpeptide N-tetradecanoyltransferase, N-terminal / Glycylpeptide N-tetradecanoyltransferase, C-terminal / Myristoyl-CoA:protein N-myristoyltransferase, N-terminal domain / Myristoyl-CoA:protein N-myristoyltransferase, C-terminal domain / Gcn5-related N-acetyltransferase (GNAT) / Acyl-CoA N-acyltransferase / Aminopeptidase / 3-Layer(aba) Sandwich / Alpha BetaSimilarity search - Domain/homology |
---|
Biological species | ![](img/tx_fungus.gif) ASPERGILLUS FUMIGATUS (mold) |
---|
Method | X-RAY DIFFRACTION / SYNCHROTRON / MOLECULAR REPLACEMENT / Resolution: 1.85 Å |
---|
Authors | Raimi, O.G. / Robinson, D.A. / Fang, W. / Blair, D.E. / Harrison, J. / Ruda, G.F. / Lockhart, D.E.A. / Torrie, L.S. / Wyatt, P.G. / Gilbert, I.H. / Van Aalten, D.M.F. |
---|
Citation | Journal: Acs Chem.Biol. / Year: 2015 Title: N-Myristoyltransferase is a Cell Wall Target in Aspergillus Fumigatus. Authors: Fang, W. / Robinson, D.A. / Raimi, O.G. / Blair, D.E. / Harrison, J.R. / Lockhart, D.E.A. / Torrie, L.S. / Ruda, G.F. / Wyatt, P.G. / Gilbert, I.H. / Van Aalten, D.M.F. |
---|
History | Deposition | Oct 9, 2013 | Deposition site: PDBE / Processing site: PDBE |
---|
Revision 1.0 | Sep 17, 2014 | Provider: repository / Type: Initial release |
---|
Revision 1.1 | Mar 23, 2016 | Group: Database references |
---|
Revision 1.2 | May 8, 2024 | Group: Data collection / Database references ...Data collection / Database references / Derived calculations / Other Category: chem_comp_atom / chem_comp_bond ...chem_comp_atom / chem_comp_bond / database_2 / pdbx_database_status / struct_site Item: _database_2.pdbx_DOI / _database_2.pdbx_database_accession ..._database_2.pdbx_DOI / _database_2.pdbx_database_accession / _pdbx_database_status.status_code_sf / _struct_site.pdbx_auth_asym_id / _struct_site.pdbx_auth_comp_id / _struct_site.pdbx_auth_seq_id |
---|
|
---|