+Search query
-Structure paper
Title | Structures of human PTP1B variants reveal allosteric sites to target for weight loss therapy |
---|---|
Journal, issue, pages | Biorxiv, Year 2024 |
Publish date | Aug 2, 2024 (structure data deposition date) |
Authors | Perdikari, A. / Woods, V. / Ebrahim, A. / Lawler, K. / Bounds, R. / Singh, N. / Mehlman, T. / Riley, B. / Sharma, S. / Morris, J. ...Perdikari, A. / Woods, V. / Ebrahim, A. / Lawler, K. / Bounds, R. / Singh, N. / Mehlman, T. / Riley, B. / Sharma, S. / Morris, J. / Keogh, J. / Henning, E. / Smith, M. / Farooqi, I. / Keedy, D. |
External links | Biorxiv / Search PubMed |
Methods | X-ray diffraction |
Resolution | 1.65 - 2.3 Å |
Structure data | PDB-9cyo: PDB-9cyp: PDB-9cyq: PDB-9cyr: |
Chemicals | ChemComp-BME: ChemComp-MG: ChemComp-HOH: |
Source |
|
Keywords | HYDROLASE / PTP1B / Phosphatase / Allostery / PTP |