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Title | Design, synthesis and biological evaluation of 5-amino-1H-pyrazole-4-carboxamide derivatives as pan-FGFR covalent inhibitors. |
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Journal, issue, pages | Eur. J. Med. Chem., Vol. 275, Page 116558-116558, Year 2024 |
Publish date | Jan 20, 2024 (structure data deposition date) |
![]() | Deng, W. / Chen, X. / Liang, H. / Song, X. / Xiang, S. / Guo, J. / Tu, Z. / Zhou, Y. / Chen, Y. / Lu, X. |
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Methods | X-ray diffraction |
Resolution | 1.75 - 2.792 Å |
Structure data | ![]() PDB-8xz7: ![]() PDB-8y22: |
Chemicals | ![]() ChemComp-SO4: ![]() PDB-1lww: ![]() ChemComp-HOH: ![]() PDB-1lw9: |
Source |
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![]() | TRANSFERASE / Fibroblast growth factor receptor 1 |