+Search query
-Structure paper
Title | Omecamtiv mecarbil and Mavacamten target the same myosin pocket despite antagonistic effects in heart contraction. |
---|---|
Journal, issue, pages | Biorxiv, Year 2023 |
Publish date | Oct 26, 2023 (structure data deposition date) |
![]() | Auguin, D. / Robert-Paganin, J. / Rety, S. / Kikuti, C. / David, A. / Theumer, G. / Schmidt, A.W. / Knolker, H.J. / Houdusse, A. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.8 - 2.759 Å |
Structure data | ![]() PDB-8qyp: ![]() PDB-8qyq: ![]() PDB-8qyr: ![]() PDB-8qyu: |
Chemicals | ![]() ChemComp-ADP: ![]() ChemComp-VO4: ![]() ChemComp-MG: ![]() ChemComp-HOH: ![]() ChemComp-BEF: ![]() ChemComp-XB2: ![]() ChemComp-FMT: ![]() ChemComp-GOL: ![]() ChemComp-SO4: ![]() ChemComp-EDO: ![]() ChemComp-DMS: ![]() ChemComp-2OW: ![]() ChemComp-MLA: |
Source |
|
![]() | CONTRACTILE PROTEIN / cardiac myosin modulators inherited cardiomyopathies / cardiac myosin modulators inherited cardiomyopathies mavcamten / cardiac myosin modulators inherited cardiomyopathies mavacamten / cardiac myosin modulators inherited cardiomyopathies Omecamtiv mecarbil |