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-Structure paper
Title | Targeting the Subpocket Enables the Discovery of Thiadiazole-Pyridazine Derivatives as Glutaminase C Inhibitors. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 14, Page 1455-1466, Year 2023 |
Publish date | Jun 26, 2023 (structure data deposition date) |
![]() | Sun, H. / Du, T. / Yang, M. / Liu, X. / Xue, X. / Chen, K. / Lang, X. / Chen, X. / Wang, B. / Wang, X. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.01 - 2.39 Å |
Structure data | ![]() PDB-8jub: ![]() PDB-8jue: |
Chemicals | ![]() ChemComp-V4I: ![]() ChemComp-HOH: ![]() ChemComp-V59: |
Source |
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![]() | HYDROLASE/HYDROLASE INHIBITOR / Inhibitor / Complex / ANTITUMOR PROTEIN / HYDROLASE-HYDROLASE INHIBITOR complex |