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-Structure paper
Title | Development of a Potent Cyclic Peptide Inhibitor of the nNOS/PSD-95 Interaction. |
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Journal, issue, pages | J. Med. Chem., Vol. 66, Page 976-990, Year 2023 |
Publish date | Nov 1, 2022 (structure data deposition date) |
Authors | Balboa, J.R. / Essig, D.J. / Ma, S. / Karer, N. / Clemmensen, L.S. / Pedersen, S.W. / Joerger, A.C. / Knapp, S. / Ostergaard, S. / Stromgaard, K. |
External links | J. Med. Chem. / PubMed:36580549 |
Methods | X-ray diffraction |
Resolution | 1.44 - 1.59 Å |
Structure data | PDB-8bi8: PDB-8bi9: |
Chemicals | ChemComp-HOH: ChemComp-TBU: |
Source |
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Keywords | PROTEIN BINDING / cyclic beta-hairpin / neuronal nitric oxidase synthase / inhibitor of the NOS/PSD-95 interaction / peptide drugs / stroke treatment |