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-Structure paper
Title | PM534, an Optimized Target-Protein Interaction Strategy through the Colchicine Site of Tubulin. |
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Journal, issue, pages | J. Med. Chem., Vol. 67, Page 2619-2630, Year 2024 |
Publish date | May 25, 2022 (structure data deposition date) |
![]() | Lucena-Agell, D. / Guillen, M.J. / Matesanz, R. / Alvarez-Bernad, B. / Hortiguela, R. / Aviles, P. / Martinez-Diez, M. / Santamaria-Nunez, G. / Contreras, J. / Plaza-Menacho, I. ...Lucena-Agell, D. / Guillen, M.J. / Matesanz, R. / Alvarez-Bernad, B. / Hortiguela, R. / Aviles, P. / Martinez-Diez, M. / Santamaria-Nunez, G. / Contreras, J. / Plaza-Menacho, I. / Gimenez-Abian, J.F. / Oliva, M.A. / Cuevas, C. / Diaz, J.F. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.45 Å |
Structure data | ![]() PDB-7zyw: |
Chemicals | ![]() ChemComp-GTP: ![]() ChemComp-GOL: ![]() ChemComp-CA: ![]() ChemComp-MG: ![]() ChemComp-CL: ![]() ChemComp-GDP: ![]() ChemComp-MES: ![]() ChemComp-KG0: ![]() ChemComp-DMS: ![]() ChemComp-ACP: ![]() ChemComp-HOH: |
Source |
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![]() | CELL CYCLE/INHIBITOR / Tubulin / microtubule destabilizing agents / inhibitor / CELL CYCLE-INHIBITOR complex |