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-Structure paper
Title | Venglustat Inhibits Protein N-Terminal Methyltransferase 1 in a Substrate-Competitive Manner. |
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Journal, issue, pages | J. Med. Chem., Vol. 65, Page 12334-12345, Year 2022 |
Publish date | Feb 21, 2022 (structure data deposition date) |
Authors | Dong, G. / Deng, Y. / Yasgar, A. / Yadav, R. / Talley, D. / Zakharov, A.V. / Jain, S. / Rai, G. / Noinaj, N. / Simeonov, A. / Huang, R. |
External links | J. Med. Chem. / PubMed:36074125 |
Methods | X-ray diffraction |
Resolution | 3.17 Å |
Structure data | PDB-7u1m: |
Chemicals | ChemComp-SAH: ChemComp-KYF: |
Source |
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Keywords | TRANSFERASE/INHIBITOR / Methyltransferase / Enzyme / Inhibitor complex / TRANSFERASE / TRANSFERASE-INHIBITOR complex |