+Search query
-Structure paper
Title | Basis for drug selectivity of plasmepsin IX and X inhibition in Plasmodium falciparum and vivax. |
---|---|
Journal, issue, pages | Structure, Vol. 30, Page 947-, Year 2022 |
Publish date | Dec 21, 2021 (structure data deposition date) |
![]() | Hodder, A.N. / Christensen, J. / Scally, S. / Triglia, T. / Ngo, A. / Birkinshaw, R.W. / Bailey, B. / Favuzza, P. / Dietrich, M.H. / Tham, W.H. ...Hodder, A.N. / Christensen, J. / Scally, S. / Triglia, T. / Ngo, A. / Birkinshaw, R.W. / Bailey, B. / Favuzza, P. / Dietrich, M.H. / Tham, W.H. / Czabotar, P.E. / Lowes, K. / Guo, Z. / Murgolo, N. / Lera Ruiz, M. / McCauley, J.A. / Sleebs, B.E. / Olsen, D. / Cowman, A.F. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.85 - 3.35 Å |
Structure data | ![]() PDB-7tbb: ![]() PDB-7tbc: ![]() PDB-7tbd: ![]() PDB-7tbe: |
Chemicals | ![]() ChemComp-NAG: ![]() ChemComp-ACT: ![]() ChemComp-GOL: ![]() ChemComp-HOH: ![]() ChemComp-EDO: ![]() ChemComp-PG4: ![]() ChemComp-I0L: ![]() ChemComp-I0I: ![]() ChemComp-SO4: |
Source |
|
![]() | HYDROLASE / Aspartyl Protease |