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-Structure paper
Title | Conformation-locking antibodies for the discovery and characterization of KRAS inhibitors. |
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Journal, issue, pages | Nat. Biotechnol., Vol. 40, Page 769-778, Year 2022 |
Publish date | Apr 5, 2021 (structure data deposition date) |
![]() | Davies, C.W. / Oh, A.J. / Mroue, R. / Steffek, M. / Bruning, J.M. / Xiao, Y. / Feng, S. / Jayakar, S. / Chan, E. / Arumugam, V. ...Davies, C.W. / Oh, A.J. / Mroue, R. / Steffek, M. / Bruning, J.M. / Xiao, Y. / Feng, S. / Jayakar, S. / Chan, E. / Arumugam, V. / Uribe, S.C. / Drummond, J. / Frommlet, A. / Lu, C. / Franke, Y. / Merchant, M. / Koeppen, H. / Quinn, J.G. / Malhotra, S. / Do, S. / Gazzard, L. / Purkey, H.E. / Rudolph, J. / Mulvihill, M.M. / Koerber, J.T. / Wang, W. / Evangelista, M. |
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Methods | X-ray diffraction |
Resolution | 1.96 - 2.2 Å |
Structure data | ![]() PDB-7mdp: ![]() PDB-7rp2: ![]() PDB-7rp3: ![]() PDB-7rp4: |
Chemicals | ![]() ChemComp-Z07: ![]() ChemComp-GDP: ![]() ChemComp-MG: ![]() ChemComp-ACT: ![]() ChemComp-CAD: ![]() ChemComp-P15: ![]() ChemComp-EDO: ![]() ChemComp-DMS: ![]() ChemComp-HOH: ![]() ChemComp-CAC: ![]() ChemComp-MKZ: ![]() ChemComp-GOL: ![]() ChemComp-SO4: |
Source |
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![]() | HYDROLASE/Immune System / KRAS / GTPase / HYDROLASE / HYDROLASE-Immune System complex / antibody / conformation-specific / inhibitor / conformation-specific antibody |