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-Structure paper
Title | Stabilization of the RAS:PDE6D Complex Is a Novel Strategy to Inhibit RAS Signaling. |
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Journal, issue, pages | J. Med. Chem., Vol. 65, Page 1898-1914, Year 2022 |
Publish date | Nov 14, 2021 (structure data deposition date) |
![]() | Yelland, T. / Garcia, E. / Parry, C. / Kowalczyk, D. / Wojnowska, M. / Gohlke, A. / Zalar, M. / Cameron, K. / Goodwin, G. / Yu, Q. ...Yelland, T. / Garcia, E. / Parry, C. / Kowalczyk, D. / Wojnowska, M. / Gohlke, A. / Zalar, M. / Cameron, K. / Goodwin, G. / Yu, Q. / Zhu, P.C. / ElMaghloob, Y. / Pugliese, A. / Archibald, L. / Jamieson, A. / Chen, Y.X. / McArthur, D. / Bower, J. / Ismail, S. |
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Methods | X-ray diffraction |
Resolution | 1.45 - 3.1 Å |
Structure data | ![]() PDB-7q9q: ![]() PDB-7q9r: ![]() PDB-7q9s: ![]() PDB-7q9u: ![]() PDB-7qf9: ![]() PDB-7qjk: |
Chemicals | ![]() ChemComp-CMT: ![]() ChemComp-EDO: ![]() ChemComp-GER: ![]() ChemComp-HOH: ![]() ChemComp-FAR: ![]() ChemComp-SO4: ![]() ChemComp-9TI: ![]() ChemComp-DMS: ![]() ChemComp-GDP: ![]() ChemComp-9VO: |
Source |
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![]() | TRANSPORT PROTEIN / Complex / PROTEIN BINDING / Inhibitor / SIGNALING PROTEIN / Cancer / Drug Discovery / trafficking / Inhibitor complex |