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-Structure paper
Title | Rational Design of Potent Inhibitors of a Metallohydrolase Using a Fragment-Based Approach. |
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Journal, issue, pages | Chemmedchem, Vol. 16, Page 3342-3359, Year 2021 |
Publish date | Jun 14, 2021 (structure data deposition date) |
Authors | Feder, D. / Mohd-Pahmi, S.H. / Hussein, W.M. / Guddat, L.W. / McGeary, R.P. / Schenk, G. |
External links | Chemmedchem / PubMed:34331400 |
Methods | X-ray diffraction |
Resolution | 2 - 2.3 Å |
Structure data | PDB-7ov2: PDB-7ov3: PDB-7ov8: |
Chemicals | ChemComp-1PE: ChemComp-P6G: ChemComp-PG4: ChemComp-GLN: ChemComp-PO4: ChemComp-EDO: ChemComp-PGE: ChemComp-GOL: ChemComp-CIT: ChemComp-NA: ChemComp-FE: ChemComp-HOH: ChemComp-DMS: ChemComp-R2J: ChemComp-NAG: ChemComp-CL: ChemComp-EPE: |
Source |
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Keywords | HYDROLASE / Purple acid phosphatase / metallohydrolases / osteoporosis / fragment-based drug design / METAL BINDING PROTEIN |