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-Structure paper
Title | Structural investigation of a pyrano-1,3-oxazine derivative and the phenanthridinone core moiety against BRD2 bromodomains. |
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Journal, issue, pages | Acta Crystallogr. ,Sect. F, Vol. 78, Page 119-127, Year 2022 |
Publish date | Apr 19, 2021 (structure data deposition date) |
![]() | Arole, A.H. / Deshmukh, P. / Sridhar, A. / Padmanabhan, B. |
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Methods | X-ray diffraction |
Resolution | 1.7 - 2.45 Å |
Structure data | ![]() PDB-7env: ![]() PDB-7enz: ![]() PDB-7eo5: |
Chemicals | ![]() ChemComp-BUX: ![]() ChemComp-SO4: ![]() ChemComp-HOH: ![]() ChemComp-LDR: ![]() ChemComp-PGE: |
Source |
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![]() | TRANSCRIPTION/INHIBITOR / BET family / BET inhibitor / Bromodomain Inhibitor / BRD2-BD1 inhibitor / TRANSCRIPTION-INHIBITOR complex / TRANSCRIPTION / BRD2 / bromodomain / b-mercaptoethanol / CME |