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-Structure paper
Title | Identification of an inhibitory pocket in falcilysin provides a new avenue for malaria drug development. |
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Journal, issue, pages | Cell Chem Biol, Vol. 31, Page 743-759.e8, Year 2024 |
Publish date | Nov 18, 2020 (structure data deposition date) |
![]() | Wirjanata, G. / Lin, J. / Dziekan, J.M. / El Sahili, A. / Chung, Z. / Tjia, S. / Binte Zulkifli, N.E. / Boentoro, J. / Tham, R. / Jia, L.S. ...Wirjanata, G. / Lin, J. / Dziekan, J.M. / El Sahili, A. / Chung, Z. / Tjia, S. / Binte Zulkifli, N.E. / Boentoro, J. / Tham, R. / Jia, L.S. / Go, K.D. / Yu, H. / Partridge, A. / Olsen, D. / Prabhu, N. / Sobota, R.M. / Nordlund, P. / Lescar, J. / Bozdech, Z. |
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Methods | X-ray diffraction |
Resolution | 1.55 - 2.003 Å |
Structure data | ![]() PDB-7di7: ![]() PDB-7dia: ![]() PDB-7dij: ![]() PDB-8ho4: ![]() PDB-8ho5: |
Chemicals | ![]() ChemComp-ACT: ![]() ChemComp-CLQ: ![]() ChemComp-ZN: ![]() ChemComp-HOH: ![]() ChemComp-H8O: ![]() ChemComp-GOL: ![]() ChemComp-YMZ: ![]() ChemComp-EDO: ![]() ChemComp-DMS: ![]() ChemComp-H8F: ![]() ChemComp-XUH: ![]() ChemComp-XUN: ![]() ChemComp-PEG: |
Source |
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![]() | PROTEIN BINDING/INHIBITOR / PROTEIN BINDING-inhibitor complex / HYDROLASE / Falcilysin / MMV000848 / Inhibitor / Complex / PROTEIN BINDING / MMV665806 |