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-Structure paper
Title | KRAS G12C fragment screening renders new binding pockets. |
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Journal, issue, pages | Small Gtpases, Vol. 13, Page 225-238, Year 2022 |
Publish date | Aug 14, 2020 (structure data deposition date) |
Authors | Mathieu, M. / Steier, V. / Fassy, F. / Delorme, C. / Papin, D. / Genet, B. / Duffieux, F. / Bertrand, T. / Delarbre, L. / Le-Borgne, H. ...Mathieu, M. / Steier, V. / Fassy, F. / Delorme, C. / Papin, D. / Genet, B. / Duffieux, F. / Bertrand, T. / Delarbre, L. / Le-Borgne, H. / Parent, A. / Didier, P. / Marquette, J.P. / Lowinski, M. / Houtmann, J. / Lamberton, A. / Debussche, L. / Alexey, R. |
External links | Small Gtpases / PubMed:34558391 |
Methods | X-ray diffraction |
Resolution | 1.32 - 2.16 Å |
Structure data | PDB-7a1w: PDB-7a1x: PDB-7a1y: PDB-7a47: |
Chemicals | ChemComp-GDP: ChemComp-MG: ChemComp-PO4: ChemComp-QWK: ChemComp-HOH: ChemComp-QWB: ChemComp-QWH: ChemComp-SO4: ChemComp-QY5: |
Source |
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Keywords | ONCOPROTEIN / inhibitor / mutant |