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-Structure paper
Title | Designed Parasite-Selective Rhomboid Inhibitors Block Invasion and Clear Blood-Stage Malaria. |
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Journal, issue, pages | Cell Chem Biol, Vol. 27, Page 1410-1424.e6, Year 2020 |
Publish date | Jan 15, 2020 (structure data deposition date) |
![]() | Gandhi, S. / Baker, R.P. / Cho, S. / Stanchev, S. / Strisovsky, K. / Urban, S. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.3 - 2.4 Å |
Structure data | ![]() PDB-6vj8: ![]() PDB-6vj9: ![]() PDB-6xro: ![]() PDB-6xrp: |
Chemicals | ![]() ChemComp-HOH: ![]() ChemComp-CL: ![]() ChemComp-NA: ![]() ChemComp-V87: |
Source |
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![]() | HYDROLASE/HYDROLASE INHIBITOR / inhibitor / complex / GlpG / rhomboid protease / HYDROLASE-HYDROLASE INHIBITOR complex / membrane protein |