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-Structure paper
Title | LipE guided discovery of isopropylphenyl pyridazines as pantothenate kinase modulators. |
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Journal, issue, pages | Bioorg. Med. Chem., Vol. 52, Page 116504-116504, Year 2021 |
Publish date | May 22, 2020 (structure data deposition date) |
![]() | Sharma, L.K. / Yun, M.K. / Subramanian, C. / Tangallapally, R. / Jackowski, S. / Rock, C.O. / White, S.W. / Lee, R.E. |
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Methods | X-ray diffraction |
Resolution | 2 - 2.3 Å |
Structure data | ![]() PDB-6x4j: ![]() PDB-6x4k: ![]() PDB-6x4l: |
Chemicals | ![]() ChemComp-MG: ![]() ChemComp-ANP: ![]() ChemComp-UOM: ![]() ChemComp-EDO: ![]() ChemComp-HOH: ![]() ChemComp-UOP: ![]() ChemComp-CL: ![]() ChemComp-UOS: |
Source |
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![]() | TRANSFERASE / PANK / Substrate / Complex / Pantothenate kinase |