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-Structure paper
Title | Structural basis for allosteric PARP-1 retention on DNA breaks. |
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Journal, issue, pages | Science, Vol. 368, Year 2020 |
Publish date | Jan 30, 2019 (structure data deposition date) |
Authors | Zandarashvili, L. / Langelier, M.F. / Velagapudi, U.K. / Hancock, M.A. / Steffen, J.D. / Billur, R. / Hannan, Z.M. / Wicks, A.J. / Krastev, D.B. / Pettitt, S.J. ...Zandarashvili, L. / Langelier, M.F. / Velagapudi, U.K. / Hancock, M.A. / Steffen, J.D. / Billur, R. / Hannan, Z.M. / Wicks, A.J. / Krastev, D.B. / Pettitt, S.J. / Lord, C.J. / Talele, T.T. / Pascal, J.M. / Black, B.E. |
External links | Science / PubMed:32241924 |
Methods | X-ray diffraction |
Resolution | 1.8 - 2.9 Å |
Structure data | PDB-6ntu: PDB-6vkk: PDB-6vko: PDB-6vkq: |
Chemicals | ChemComp-DMS: ChemComp-1PE: ChemComp-L1S: ChemComp-SO4: ChemComp-HOH: ChemComp-RPB: ChemComp-GOL: ChemComp-UHB: |
Source |
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Keywords | transferase/transferase inhibitor / PARP-1 / poly(ADP-ribose) polymerase / PARP inhibitor / PARP1 / ARTD1 / TRANSFERASE / transferase-transferase inhibitor complex / TRANSFERASE/INHIBITOR / TRANSFERASE-INHIBITOR complex |