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-Structure paper
Title | Pharmacological chaperones for GCase that switch conformation with pH enhance enzyme levels in Gaucher animal models. |
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Journal, issue, pages | To Be Published |
Publish date | Aug 5, 2019 (structure data deposition date) |
![]() | Santana, A.G. / Robinson, K. / Vickers, C. / Chen, H. / Zhou, S. / Boraston, A.B. / Clarke, L.A. / Withers, S.G. |
![]() | Search PubMed |
Methods | X-ray diffraction |
Resolution | 2.526 - 2.796 Å |
Structure data | ![]() PDB-6q1n: ![]() PDB-6q1p: |
Chemicals | ![]() ChemComp-EDO: ![]() ChemComp-SO4: ![]() ChemComp-P9V: ![]() ChemComp-NAG: ![]() ChemComp-HOH: ![]() ChemComp-P8Y: |
Source |
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![]() | HYDROLASE/INHIBITOR / pharmacological chaperone / Gaucher disease / glycosidase / inhibitor / pKa / HYDROLASE / HYDROLASE-INHIBITOR complex |