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-Structure paper
Title | Novel Propargyl-Linked Bisubstrate Analogues as Tight-Binding Inhibitors for NicotinamideN-Methyltransferase. |
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Journal, issue, pages | J. Med. Chem., Vol. 62, Page 10783-10797, Year 2019 |
Publish date | Jul 20, 2019 (structure data deposition date) |
Authors | Chen, D. / Li, L. / Diaz, K. / Iyamu, I.D. / Yadav, R. / Noinaj, N. / Huang, R. |
External links | J. Med. Chem. / PubMed:31724854 |
Methods | X-ray diffraction |
Resolution | 2.3 - 2.575 Å |
Structure data | PDB-6pve: PDB-6pvs: |
Chemicals | ChemComp-OZP: ChemComp-HOH: ChemComp-P0V: |
Source |
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Keywords | TRANSFERASE/TRANSFERASE Inhibitor / Methyltransferase / Inhibitor / TRANSFERASE / TRANSFERASE-TRANSFERASE Inhibitor complex |