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Title | Targeting the PI5P4K Lipid Kinase Family in Cancer Using Covalent Inhibitors. |
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Journal, issue, pages | Cell Chem Biol, Vol. 27, Page 525-, Year 2020 |
Publish date | May 1, 2019 (structure data deposition date) |
Authors | Sivakumaren, S.C. / Shim, H. / Zhang, T. / Ferguson, F.M. / Lundquist, M.R. / Browne, C.M. / Seo, H.S. / Paddock, M.N. / Manz, T.D. / Jiang, B. ...Sivakumaren, S.C. / Shim, H. / Zhang, T. / Ferguson, F.M. / Lundquist, M.R. / Browne, C.M. / Seo, H.S. / Paddock, M.N. / Manz, T.D. / Jiang, B. / Hao, M.F. / Krishnan, P. / Wang, D.G. / Yang, T.J. / Kwiatkowski, N.P. / Ficarro, S.B. / Cunningham, J.M. / Marto, J.A. / Dhe-Paganon, S. / Cantley, L.C. / Gray, N.S. |
External links | Cell Chem Biol / PubMed:32130941 |
Methods | X-ray diffraction |
Resolution | 2.21 Å |
Structure data | PDB-6osp: |
Chemicals | ChemComp-N51: ChemComp-GOL: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE / kinase / SIGNALING PROTEIN |