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-Structure paper
Title | Discovery of a chemical probe for PRDM9. |
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Journal, issue, pages | Nat Commun, Vol. 10, Page 5759-5759, Year 2019 |
Publish date | Jan 10, 2019 (structure data deposition date) |
![]() | Allali-Hassani, A. / Szewczyk, M.M. / Ivanochko, D. / Organ, S.L. / Bok, J. / Ho, J.S.Y. / Gay, F.P.H. / Li, F. / Blazer, L. / Eram, M.S. ...Allali-Hassani, A. / Szewczyk, M.M. / Ivanochko, D. / Organ, S.L. / Bok, J. / Ho, J.S.Y. / Gay, F.P.H. / Li, F. / Blazer, L. / Eram, M.S. / Halabelian, L. / Dilworth, D. / Luciani, G.M. / Lima-Fernandes, E. / Wu, Q. / Loppnau, P. / Palmer, N. / Talib, S.Z.A. / Brown, P.J. / Schapira, M. / Kaldis, P. / O'Hagan, R.C. / Guccione, E. / Barsyte-Lovejoy, D. / Arrowsmith, C.H. / Sanders, J.M. / Kattar, S.D. / Bennett, D.J. / Nicholson, B. / Vedadi, M. |
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Methods | X-ray diffraction |
Resolution | 2.58 Å |
Structure data | ![]() PDB-6nm4: |
Chemicals | ![]() ChemComp-ZN: ![]() ChemComp-SAM: ![]() ChemComp-KS7: ![]() ChemComp-UNX: ![]() ChemComp-HOH: |
Source |
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![]() | GENE REGULATION/INHIBITOR / PR SET domain / Lysine Methyltransferase / Inhibitor / Structural Genomics / Structural Genomics Consortium / SGC / GENE REGULATION-INHIBITOR complex |