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-Structure paper
Title | Discovery of a dual inhibitor of NQO1 and GSTP1 for treating glioblastoma. |
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Journal, issue, pages | J Hematol Oncol, Vol. 13, Page 141-141, Year 2020 |
Publish date | Dec 23, 2019 (structure data deposition date) |
![]() | Lei, K. / Gu, X. / Alvarado, A.G. / Du, Y. / Luo, S. / Ahn, E.H. / Kang, S.S. / Ji, B. / Liu, X. / Mao, H. ...Lei, K. / Gu, X. / Alvarado, A.G. / Du, Y. / Luo, S. / Ahn, E.H. / Kang, S.S. / Ji, B. / Liu, X. / Mao, H. / Fu, H. / Kornblum, H.I. / Jin, L. / Li, H. / Ye, K. |
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Methods | X-ray diffraction |
Resolution | 1.581 - 2.501 Å |
Structure data | ![]() PDB-6llc: ![]() PDB-6llx: |
Chemicals | ![]() ChemComp-FAD: ![]() ChemComp-EHL: ![]() ChemComp-SO4: ![]() ChemComp-HOH: ![]() ChemComp-GSH: ![]() ChemComp-MES: |
Source |
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![]() | OXIDOREDUCTASE / Oxidative stress / GBM / small molecular inhibitor / TRANSFERASE / NQO1 / GSTP1 |