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-Structure paper
Title | Aiming to Miss a Moving Target: Bromo and Extra Terminal Domain (BET) Selectivity in Constrained ATAD2 Inhibitors. |
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Journal, issue, pages | J. Med. Chem., Vol. 61, Page 8321-8336, Year 2018 |
Publish date | Aug 18, 2018 (structure data deposition date) |
Authors | Bamborough, P. / Chung, C.W. / Furze, R.C. / Grandi, P. / Michon, A.M. / Watson, R.J. / Mitchell, D.J. / Barnett, H. / Prinjha, R.K. / Rau, C. ...Bamborough, P. / Chung, C.W. / Furze, R.C. / Grandi, P. / Michon, A.M. / Watson, R.J. / Mitchell, D.J. / Barnett, H. / Prinjha, R.K. / Rau, C. / Sheppard, R.J. / Werner, T. / Demont, E.H. |
External links | J. Med. Chem. / PubMed:30226378 |
Methods | X-ray diffraction |
Resolution | 1.7 - 2.61 Å |
Structure data | PDB-6hdn: PDB-6hdo: PDB-6hdq: |
Chemicals | ChemComp-SO4: ChemComp-EDO: ChemComp-FZB: ChemComp-HOH: ChemComp-FZH: ChemComp-FZE: |
Source |
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Keywords | TRANSCRIPTION / INHIBITOR / ATAD2 / BROMODOMAIN / EPIGENETICS / ATPase family AAA domain-containing protein 2 / HISTONE / EPIGENETIC READER / BRD4 / BROMODOMAIN CONTAINING PROTEIN 4 / ANTAGONIST |