+Search query
-Structure paper
Title | Covalent Docking Identifies a Potent and Selective MKK7 Inhibitor. |
---|---|
Journal, issue, pages | Cell Chem Biol, Vol. 26, Page 98-108.e5, Year 2019 |
Publish date | Dec 26, 2017 (structure data deposition date) |
Authors | Shraga, A. / Olshvang, E. / Davidzohn, N. / Khoshkenar, P. / Germain, N. / Shurrush, K. / Carvalho, S. / Avram, L. / Albeck, S. / Unger, T. ...Shraga, A. / Olshvang, E. / Davidzohn, N. / Khoshkenar, P. / Germain, N. / Shurrush, K. / Carvalho, S. / Avram, L. / Albeck, S. / Unger, T. / Lefker, B. / Subramanyam, C. / Hudkins, R.L. / Mitchell, A. / Shulman, Z. / Kinoshita, T. / London, N. |
External links | Cell Chem Biol / PubMed:30449673 |
Methods | X-ray diffraction |
Resolution | 2.28 - 2.3 Å |
Structure data | PDB-5z1d: PDB-5z1e: |
Chemicals | ChemComp-95U: ChemComp-EPE: ChemComp-HOH: |
Source |
|
Keywords | TRANSFERASE / protein kinase |