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-Structure paper
Title | Crystal Structures of Spleen Tyrosine Kinase in Complex with Two Novel 4-Aminopyrido[4,3-d] Pyrimidine Derivative Inhibitors. |
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Journal, issue, pages | Mol. Cells, Vol. 41, Page 545-552, Year 2018 |
Publish date | Aug 9, 2017 (structure data deposition date) |
![]() | Lee, S.J. / Choi, J.S. / Bong, S.M. / Hwang, H.J. / Lee, J. / Song, H.J. / Kim, J.H. / Koh, J.S. / Lee, B.I. |
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Methods | X-ray diffraction |
Resolution | 1.8 - 2.14 Å |
Structure data | ![]() PDB-5y5t: ![]() PDB-5y5u: |
Chemicals | ![]() ChemComp-8OR: ![]() ChemComp-HOH: ![]() ChemComp-8OU: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / Inhibitor / Spleen Tyrosine Kinase / human kinase / drug discovery / TRANSFERASE / TRANSFERASE-TRANSFERASE INHIBITOR complex |