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-Structure paper
Title | Structure-activity relationship studies of G9a-like protein (GLP) inhibitors. |
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Journal, issue, pages | Bioorg. Med. Chem., Vol. 25, Page 4414-4423, Year 2017 |
Publish date | May 11, 2017 (structure data deposition date) |
Authors | Xiong, Y. / Li, F. / Babault, N. / Wu, H. / Dong, A. / Zeng, H. / Chen, X. / Arrowsmith, C.H. / Brown, P.J. / Liu, J. ...Xiong, Y. / Li, F. / Babault, N. / Wu, H. / Dong, A. / Zeng, H. / Chen, X. / Arrowsmith, C.H. / Brown, P.J. / Liu, J. / Vedadi, M. / Jin, J. |
External links | Bioorg. Med. Chem. / PubMed:28662962 |
Methods | X-ray diffraction |
Resolution | 1.4 - 1.85 Å |
Structure data | PDB-5vsc: PDB-5vsd: PDB-5vse: PDB-5vsf: |
Chemicals | ChemComp-ZN: ChemComp-SAM: ChemComp-9HJ: ChemComp-HOH: ChemComp-DIO: ChemComp-GOL: ChemComp-9HG: |
Source |
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Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / protein-small molecule inhibitor complex / TRANSFERASE-TRANSFERASE INHIBITOR complex |