+Search query
-Structure paper
Title | Discovery and Characterization of Allosteric WNK Kinase Inhibitors. |
---|---|
Journal, issue, pages | ACS Chem. Biol., Vol. 11, Page 3338-3346, Year 2016 |
Publish date | Sep 24, 2016 (structure data deposition date) |
Authors | Yamada, K. / Zhang, J.H. / Xie, X. / Reinhardt, J. / Xie, A.Q. / LaSala, D. / Kohls, D. / Yowe, D. / Burdick, D. / Yoshisue, H. ...Yamada, K. / Zhang, J.H. / Xie, X. / Reinhardt, J. / Xie, A.Q. / LaSala, D. / Kohls, D. / Yowe, D. / Burdick, D. / Yoshisue, H. / Wakai, H. / Schmidt, I. / Gunawan, J. / Yasoshima, K. / Yue, Q.K. / Kato, M. / Mogi, M. / Idamakanti, N. / Kreder, N. / Drueckes, P. / Pandey, P. / Kawanami, T. / Huang, W. / Yagi, Y.I. / Deng, Z. / Park, H.M. |
External links | ACS Chem. Biol. / PubMed:27712055 |
Methods | X-ray diffraction |
Resolution | 2.5 Å |
Structure data | PDB-5tf9: |
Chemicals | ChemComp-7AV: ChemComp-ANP: ChemComp-MN: ChemComp-CA: ChemComp-HOH: |
Source |
|
Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / Serine-threonine-protein kinase / inhibitor / ternary / complex / allosteric / TRANSFERASE-TRANSFERASE INHIBITOR complex |