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-Structure paper
Title | Structures of Human A1 and A2A Adenosine Receptors with Xanthines Reveal Determinants of Selectivity. |
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Journal, issue, pages | Structure, Vol. 25, Page 1275-1285.e4, Year 2017 |
Publish date | Jan 31, 2017 (structure data deposition date) |
![]() | Cheng, R.K.Y. / Segala, E. / Robertson, N. / Deflorian, F. / Dore, A.S. / Errey, J.C. / Fiez-Vandal, C. / Marshall, F.H. / Cooke, R.M. |
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Methods | X-ray diffraction |
Resolution | 2 - 3.303 Å |
Structure data | ![]() PDB-5mzj: ![]() PDB-5mzp: ![]() PDB-5n2r: ![]() PDB-5n2s: |
Chemicals | ![]() ChemComp-NA: ![]() ChemComp-TEP: ![]() ChemComp-CLR: ![]() ChemComp-OLA: ![]() ChemComp-OLC: ![]() ChemComp-HOH: ![]() ChemComp-CFF: ![]() ChemComp-TAR: ![]() ChemComp-8JN: ![]() ChemComp-8K8: ![]() ChemComp-SO4: |
Source |
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![]() | MEMBRANE PROTEIN / G-PROTEIN-COUPLED RECEPTOR / INTEGRAL THERMOSTABILIZING MUTATIONS / INTEGRAL MEMBRANE PROTEIN / CHIMERA / THERMOSTABILIZING MUTATIONS |