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-Structure paper
Title | Dual protein kinase and nucleoside kinase modulators for rationally designed polypharmacology. |
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Journal, issue, pages | Nat Commun, Vol. 8, Page 1420-1420, Year 2017 |
Publish date | Dec 20, 2016 (structure data deposition date) |
Authors | Hammam, K. / Saez-Ayala, M. / Rebuffet, E. / Gros, L. / Lopez, S. / Hajem, B. / Humbert, M. / Baudelet, E. / Audebert, S. / Betzi, S. ...Hammam, K. / Saez-Ayala, M. / Rebuffet, E. / Gros, L. / Lopez, S. / Hajem, B. / Humbert, M. / Baudelet, E. / Audebert, S. / Betzi, S. / Lugari, A. / Combes, S. / Letard, S. / Casteran, N. / Mansfield, C. / Moussy, A. / De Sepulveda, P. / Morelli, X. / Dubreuil, P. |
External links | Nat Commun / PubMed:29127277 |
Methods | X-ray diffraction |
Resolution | 3.2 - 3.7 Å |
Structure data | PDB-5mqj: PDB-5mql: PDB-5mqt: |
Chemicals | ChemComp-UDP: ChemComp-UMP: ChemComp-MG: ChemComp-G65: ChemComp-DCM: ChemComp-HOH: ChemComp-STI: |
Source |
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Keywords | TRANSFERASE / Deoxycytidine kinase / dCK / masitinib |