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-Structure paper
Title | Inhibitors of PEX14 disrupt protein import into glycosomes and kill Trypanosoma parasites. |
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Journal, issue, pages | Science, Vol. 355, Page 1416-1420, Year 2017 |
Publish date | Jun 7, 2016 (structure data deposition date) |
![]() | Dawidowski, M. / Emmanouilidis, L. / Kalel, V.C. / Tripsianes, K. / Schorpp, K. / Hadian, K. / Kaiser, M. / Maser, P. / Kolonko, M. / Tanghe, S. ...Dawidowski, M. / Emmanouilidis, L. / Kalel, V.C. / Tripsianes, K. / Schorpp, K. / Hadian, K. / Kaiser, M. / Maser, P. / Kolonko, M. / Tanghe, S. / Rodriguez, A. / Schliebs, W. / Erdmann, R. / Sattler, M. / Popowicz, G.M. |
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Methods | X-ray diffraction / NMR (solution) |
Resolution | 0.87 - 1.57 Å |
Structure data | ![]() PDB-5l87: ![]() PDB-5l8a: ![]() PDB-5mmc: ![]() PDB-5n8v: |
Chemicals | ![]() ChemComp-6RD: ![]() ChemComp-EDO: ![]() ChemComp-HOH: ![]() ChemComp-6RB: ![]() ChemComp-GLY: ![]() ChemComp-NA: ![]() ChemComp-KZZ: ![]() ChemComp-SO4: ![]() ChemComp-BME: ![]() ChemComp-CL: |
Source |
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![]() | MEMBRANE PROTEIN / trypanosomiasis / glycosome / protein-protein interaction inhibitor / structure-based drug discovery / inhibitor / SIGNALING PROTEIN / Peroxin 14 / Pex14 / Trypanosoma / peroxisome |