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-Structure paper
Title | Potent and Selective BACE-1 Peptide Inhibitors Lower Brain A beta Levels Mediated by Brain Shuttle Transport. |
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Journal, issue, pages | EBioMedicine, Vol. 24, Page 76-92, Year 2017 |
Publish date | Nov 9, 2016 (structure data deposition date) |
![]() | Ruderisch, N. / Schlatter, D. / Kuglstatter, A. / Guba, W. / Huber, S. / Cusulin, C. / Benz, J. / Rufer, A.C. / Hoernschemeyer, J. / Schweitzer, C. ...Ruderisch, N. / Schlatter, D. / Kuglstatter, A. / Guba, W. / Huber, S. / Cusulin, C. / Benz, J. / Rufer, A.C. / Hoernschemeyer, J. / Schweitzer, C. / Bulau, T. / Gartner, A. / Hoffmann, E. / Niewoehner, J. / Patsch, C. / Baumann, K. / Loetscher, H. / Kitas, E. / Freskgard, P.O. |
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Methods | X-ray diffraction |
Resolution | 1.82 - 2.95 Å |
Structure data | ![]() PDB-5mbw: ![]() PDB-5mco: ![]() PDB-5mcq: |
Chemicals | ![]() ChemComp-CL: ![]() ChemComp-HOH: ![]() ChemComp-BSD: ![]() ChemComp-EDO: |
Source |
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![]() | HYDROLASE / PROTEASE INHIBITOR / HYDROLASE-HYDROLASE INHIBITOR COMPLEX / EXOSITE |