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TitleIdentification of potent and selective retinoic acid receptor gamma (RAR gamma ) antagonists for the treatment of osteoarthritis pain using structure based drug design.
Journal, issue, pagesBioorg. Med. Chem. Lett., Vol. 26, Page 3274-3277, Year 2016
Publish dateMay 17, 2016 (structure data deposition date)
AuthorsHughes, N.E. / Bleisch, T.J. / Jones, S.A. / Richardson, T.I. / Doti, R.A. / Wang, Y. / Stout, S.L. / Durst, G.L. / Chambers, M.G. / Oskins, J.L. ...Hughes, N.E. / Bleisch, T.J. / Jones, S.A. / Richardson, T.I. / Doti, R.A. / Wang, Y. / Stout, S.L. / Durst, G.L. / Chambers, M.G. / Oskins, J.L. / Lin, C. / Adams, L.A. / Page, T.J. / Barr, R.J. / Zink, R.W. / Osborne, H. / Montrose-Rafizadeh, C. / Norman, B.H.
External linksBioorg. Med. Chem. Lett. / PubMed:27261179
MethodsX-ray diffraction
Resolution1.85 Å
Structure data

PDB-5k13:
Crystal structure of the RAR alpha ligand-binding domain in complex with an antagonist
Method: X-RAY DIFFRACTION / Resolution: 1.85 Å

Chemicals

ChemComp-6Q7:
4-{5-(3-tert-butylphenyl)-1-[4-(methylsulfonyl)phenyl]-1H-pyrazol-3-yl}benzoic acid

ChemComp-HOH:
WATER

Source
  • homo sapiens (human)
KeywordsTRANSCRIPTION / NHR ligand-binding domain / antagonist

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