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Title | The EED protein-protein interaction inhibitor A-395 inactivates the PRC2 complex. |
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Journal, issue, pages | Nat. Chem. Biol., Vol. 13, Page 389-395, Year 2017 |
Publish date | May 17, 2016 (structure data deposition date) |
Authors | He, Y. / Selvaraju, S. / Curtin, M.L. / Jakob, C.G. / Zhu, H. / Comess, K.M. / Shaw, B. / The, J. / Lima-Fernandes, E. / Szewczyk, M.M. ...He, Y. / Selvaraju, S. / Curtin, M.L. / Jakob, C.G. / Zhu, H. / Comess, K.M. / Shaw, B. / The, J. / Lima-Fernandes, E. / Szewczyk, M.M. / Cheng, D. / Klinge, K.L. / Li, H.Q. / Pliushchev, M. / Algire, M.A. / Maag, D. / Guo, J. / Dietrich, J. / Panchal, S.C. / Petros, A.M. / Sweis, R.F. / Torrent, M. / Bigelow, L.J. / Senisterra, G. / Li, F. / Kennedy, S. / Wu, Q. / Osterling, D.J. / Lindley, D.J. / Gao, W. / Galasinski, S. / Barsyte-Lovejoy, D. / Vedadi, M. / Buchanan, F.G. / Arrowsmith, C.H. / Chiang, G.G. / Sun, C. / Pappano, W.N. |
External links | Nat. Chem. Biol. / PubMed:28135237 |
Methods | X-ray diffraction |
Resolution | 1.83 Å |
Structure data | PDB-5k0m: |
Chemicals | ChemComp-6PU: ChemComp-HOH: |
Source |
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Keywords | PROTEIN BINDING / WD40 PRC2 |