+Search query
-Structure paper
Title | Structure-guided design of novel Trypanosoma brucei Methionyl-tRNA synthetase inhibitors. |
---|---|
Journal, issue, pages | Eur J Med Chem, Vol. 124, Page 1081-1092, Year 2016 |
Publish date | Apr 1, 2016 (structure data deposition date) |
![]() | Huang, W. / Zhang, Z. / Barros-Alvarez, X. / Koh, C.Y. / Ranade, R.M. / Gillespie, J.R. / Creason, S.A. / Shibata, S. / Verlinde, C.L. / Hol, W.G. ...Huang, W. / Zhang, Z. / Barros-Alvarez, X. / Koh, C.Y. / Ranade, R.M. / Gillespie, J.R. / Creason, S.A. / Shibata, S. / Verlinde, C.L. / Hol, W.G. / Buckner, F.S. / Fan, E. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.4 - 2.8 Å |
Structure data | ![]() PDB-5j58: ![]() PDB-5j59: ![]() PDB-5j5a: |
Chemicals | ![]() ChemComp-MET: ![]() ChemComp-GOL: ![]() ChemComp-DMS: ![]() ChemComp-N56: ![]() ChemComp-HOH: ![]() ChemComp-N93: ![]() ChemComp-756: |
Source |
|
![]() | Ligase/Ligase Inhibitor / synthetase / ligase / methionine / inhibitor / Ligase-Ligase Inhibitor complex |