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-Structure paper
Title | Development and crystallographic evaluation of histone H3 peptide with N-terminal serine substitution as a potent inhibitor of lysine-specific demethylase 1. |
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Journal, issue, pages | Bioorg. Med. Chem., Vol. 25, Page 2617-2624, Year 2017 |
Publish date | Nov 14, 2016 (structure data deposition date) |
![]() | Amano, Y. / Kikuchi, M. / Sato, S. / Yokoyama, S. / Umehara, T. / Umezawa, N. / Higuchi, T. |
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Methods | X-ray diffraction |
Resolution | 2.53 - 2.69 Å |
Structure data | ![]() PDB-5h6q: ![]() PDB-5h6r: ![]() PDB-5x60: |
Chemicals | ![]() ChemComp-GOL: ![]() ChemComp-FAD: ![]() ChemComp-HOH: |
Source |
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![]() | OXIDOREDUCTASE/TRANSCRIPTION/INHIBITOR / DEMETHYLASE / AMINE OXIDASE / CHROMATIN / HISTONE / FAD / COREPRESSOR / OXIDOREDUCTASE-TRANSCRIPTION-INHIBITOR complex / OXIDOREDUCTASE/TRANSCRIPTION / OXIDOREDUCTASE-TRANSCRIPTION complex |