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-Structure paper
Title | The polar warhead of a TRIM24 bromodomain inhibitor rearranges a water-mediated interaction network |
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Journal, issue, pages | FEBS J., Vol. 284, Page 1082-1095, Year 2017 |
Publish date | Oct 11, 2016 (structure data deposition date) |
![]() | Liu, J. / Li, F. / Bao, H. / Jiang, Y. / Zhang, S. / Ma, R. / Gao, J. / Wu, J. / Ruan, K. |
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Methods | X-ray diffraction |
Resolution | 1.901 - 2.002 Å |
Structure data | ![]() PDB-5h1t: ![]() PDB-5h1u: ![]() PDB-5h1v: |
Chemicals | ![]() ChemComp-ZN: ![]() ChemComp-7FF: ![]() ChemComp-DMS: ![]() ChemComp-HOH: ![]() ChemComp-6KT: ![]() ChemComp-7FU: |
Source |
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![]() | TRANSCRIPTION/TRANSCRIPTION INHIBITOR / TRANSCRIPTION / TRANSCRIPTION INHIBITOR / TRANSCRIPTION-TRANSCRIPTION INHIBITOR complex / TRANSCRIPTION TRANSCRIPTION INHIBITOR |